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modulátory GABA
Č. záznamu d018757 Dátum 06.06.2025 Typ M Tematický termín modulátory GABA Iný termín Angličtina (Pseudonym) gamma-Aminobutyric Acid Modulators
Slovenčina (Pseudonym) modulátory kyseliny gama maslovej
Pozri tiež (Skutočné meno) hypnotiká a sedatíva
(Skutočné meno) anxiolytiká
(Skutočné meno) anestetiká celkové
(Novšie záhlavie) GABA transportné proteíny plazmatickej membrány
MDT D27.505.519.625.240.500D27.505.696.577.240.500 Poznámka Substances that do not act as agonists or antagonists but do affect the GAMMA-AMINOBUTYRIC ACID receptor-ionophore complex. GABA-A receptors (RECEPTORS, GABA-A) appear to have at least three allosteric sites at which modulators act: a site at which BENZODIAZEPINES act by increasing the opening frequency of GAMMA-AMINOBUTYRIC ACID-activated chloride channels; a site at which BARBITURATES act to prolong the duration of channel opening; and a site at which some steroids may act. GENERAL ANESTHETICS probably act at least partly by potentiating GABAergic responses, but they are not included here. predmetové heslo
Počet záznamov: 1